Tirzepatide - Tirzepatide is a 39-amino-acid peptide with dual agonist act
Bestseller

Tirzepatide

5.0 (7)

Tirzepatide is a 39-amino-acid peptide with dual agonist activity at the GIP and GLP-1 receptors. Research compound, supplied as lyophilised powder.

MetabolicEndocrine
In Stock

1 vial · 10 mg total

Checking availability…

Total Price

฿2200

VisaMastercardApple PayKlarnaiDEALBitcoinUSDT& more more: Bancontact, Open Banking, Cash App, Afterpay, more coinsCrypto −5%Encrypted checkout

For research & laboratory use only. Not for human consumption.

Shipping: free within Thailand, ฿700 worldwide. Added at checkout. Delivery times & countries

Half-Life

5 days

Metabolic Endpoints

HbA1c and lipid endpoints reported in the trial literature

Five-Day Half-Life

C20 fatty-diacid moiety with albumin binding

DPP-4 Resistant

Aib substitutions at positions 2 and 13

Mechanism of Action

Tirzepatide is a single peptide with agonist activity at two incretin receptors, glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1). Both are class B G-protein coupled receptors signalling through cAMP. The molecule carries a C20 fatty-diacid moiety that promotes reversible albumin binding, giving a plasma half-life of roughly five days. Its receptor selectivity is biased towards GIP relative to GLP-1.

Scientific Research

Why Researchers Choose Tirzepatide

Tirzepatide (the GLP-1 and GIP dual agonist marketed as Mounjaro) is studied wherever combined incretin receptor pharmacology matters:

  • Dual incretin receptor pharmacology and additive GIP plus GLP-1 engagement studies
  • Incretin receptor signalling in hypothalamic and pancreatic tissue
  • Glycaemic control and insulin-sensitivity studies in insulin-resistant research models
  • Lipid metabolism and adipose-tissue remodelling investigations
  • Comparative pharmacology against single-receptor GLP-1 agonists such as semaglutide
  • Cardiovascular and metabolic risk-marker modulation in metabolic disease contexts

How Tirzepatide Works

Tirzepatide is a single 39-amino-acid peptide engineered to activate two incretin receptors at once: GLP-1 and GIP. A fatty-acid chain enables albumin binding for a roughly five-day half-life. GLP-1 receptor activation drives glucose-dependent insulin secretion, suppresses glucagon, slows gastric emptying and reduces appetite, while added GIP receptor engagement further enhances the insulin response and influences adipose-tissue metabolism. The combined action on both pathways is what produced larger weight and glucose effects than single-receptor GLP-1 agonists in clinical trials.

Tirzepatide vs. Semaglutide

Tirzepatide is a GLP-1 and GIP dual agonist, whereas semaglutide targets GLP-1 alone and retatrutide adds a third (glucagon) receptor. Comparing single-, dual- and triple-receptor pharmacology is a central theme in current incretin research. See the semaglutide vs. tirzepatide comparison for a side-by-side breakdown.

Reconstitution and Storage

Reconstitution: use bacteriostatic water (1 to 2ml per vial); swirl gently until fully dissolved, do not shake. After reconstitution: keep refrigerated, use within 28 days, and protect from direct light.

Vial & calculation

Calculate concentration and volume from the labelled amount, your final solution volume and a target amount you provide.

Open calculator for Tirzepatide

Current product variants are listed in the calculator. No personal dose is selected for you.

Product FAQs

Customer Reviews

5.0 (7)

Fairly easy system, decent price.

Nanak Verified
2026-09-23

Real and works very good

Ollie Verified
2026-08-31

help to reduce appetite, increase fullness, and improve blood sugar control. good for weight loss but should talk with a healthcare professional.

Elixa Verified
2026-08-25

I recently started Milo-Lab's Tirzepatide after allowing myself to blow out over 15kg from my ideal body weight, and needed to get back into shape and overhaul my diet. I'm currently in Week 3, so it's early to post a review, but the results so far have been extraordinary, so I thought it might help others considering their own weight loss journey. My results so far: Starting weight: 99.80kg Week 1: 94.80kg (5kg loss) Week 2: 92.70kg (7.1kg loss) Week 3: 90.30kg (9.50kg loss) I started with a 48hr fast, and since then my diet has been 99% keto, with a little chocolate after dinner. My training is 5 x 10km runs while fasted in the morning. Zero side effects, and this product has allowed me to properly address my diet and eat clean without much effort. I've been a long-time customer of Milo-Lab, and after listening to Matt's recommendation, I'm absolutely delighted with this product and the results. Worth every cent and more.

Anton L.
2026-02-13

Fantastic quality! Fast shipping and excellent service!

Johanna P.
2025-02-21

I tried 2.5mg and the dose feels pretty on point compared to other lab-tested Tirzepatide products I've run before. No hunger whatsoever for a couple of days!

Felix R.
2024-12-05

Game changer, the best product on the market for weight loss!

Marco P.
2024-12-01

Used in Research Stacks

GLP-1 Receptor Blend

Tirzepatide
View Stack Research

Related Products