Bremelanotide PT-141
What is Bremelanotide PT-141?
PT-141, also known as Bremelanotide, is a synthetic peptide that is used to treat sexual dysfunction in
men and women. While Viagra and Cialis, which are PDE-5 inhibitors that work to increase blood flow
into the penis, PT-141 is a melanocortin, which works at the brain to increase sexual desire. The synthetic
peptide blend was developed from Melanotan II, and was originally intended to darken skin pigmentation
and induce tanning. However, during the initial testing, patients noted a pleasant side effect – that it
caused increased sexual arousal.
How Does Bremelanotide PT-141 Work?
Bremelanotide PT-141 is a molecule that binds to and activates the melanocortin receptors associated with
skin pigmentation. Being that it
Currently, Bremelanotide PT-141 is administered via a subcutaneous injection, ideally where there are fat
deposits. The only legitimate form of the peptide is injectable. Oral pills, nasal sprays, and creams have
not been shown to be an effective means in which to administer Bremelanotide PT-141.
Given that everyone responds differently to Bremelanotide PT-141, effective dosages may vary. A 2mg
dose is generally effective for men and women, about 1 hour prior to sexual activity. Some studies suggest
starting with a 1mg test dose and injecting an identical amount 30 minutes later. By consulting your
Men’s Health Institute physician, you can receive a cycle protocol best suited for your condition. In
studies, some subjects responded to PT-141 in minutes while others took several hours to see the effects.
Bremelanotide PT-141 is a novel treatment option for sexual dysfunction that works in both men and
women.